{"id":39176,"date":"2017-12-12T00:00:00","date_gmt":"2017-12-11T23:00:00","guid":{"rendered":"http:\/\/www.pcb.ub.edu\/\/cerco-al-cancer-de-prostata-avanzado\/"},"modified":"2020-11-16T16:22:56","modified_gmt":"2020-11-16T15:22:56","slug":"cerco-al-cancer-de-prostata-avanzado","status":"publish","type":"post","link":"https:\/\/www.pcb.ub.edu\/es\/cerco-al-cancer-de-prostata-avanzado\/","title":{"rendered":"Cerco al c\u00e1ncer de pr\u00f3stata avanzado"},"content":{"rendered":"<p>En la mayor\u00eda de los casos, el c\u00e1ncer de pr\u00f3stata se cura extirpando el tumor con cirug\u00eda y\/o con radioterapia. Sin embargo, hay un 20% de pacientes que necesitar\u00e1n tratamiento para eliminar c\u00e9lulas tumorales pero, inevitablemente, deja de funcionar despu\u00e9s de dos o tres a\u00f1os y el c\u00e1ncer progresa. En este estadio de la enfermedad, ya no hay cura.\u00a0<\/p>\n<p>Las c\u00e9lulas tumorales de pr\u00f3stata necesitan que la prote\u00edna receptor de andr\u00f3genos est\u00e9 muy activa para sobrevivir y proliferar. El f\u00e1rmaco que se usa para eliminar las c\u00e9lulas tumorales interfiere, de hecho, con esta prote\u00edna. El f\u00e1rmaco act\u00faa uni\u00e9ndose a una regi\u00f3n concreta del receptor de andr\u00f3genos e inhabilita la prote\u00edna.\u00a0\u00abCon el tiempo la prote\u00edna acumula alteraciones, muta, y llega un momento en que es in\u00fatil enviar f\u00e1rmacos a aquella regi\u00f3n, porque de hecho, la prote\u00edna se desprende de esa parte\u00bb,\u00a0describe\u00a0\u00a0Xavier Salvatella.<\/p>\n<p>En el\u00a0<a href=\"https:\/\/www.irbbarcelona.org\/es\/research\/laboratory-of-molecular-biophysics\" target=\"_blank\" rel=\"noopener noreferrer\">Laboratorio en Biof\u00edsica Molecular<\/a>\u00a0dirigido por\u00a0Salvatella\u00a0estudian en detalle la estructura tridimensional y los movimientos at\u00f3micos del receptor de andr\u00f3genos para encontrar nuevos puntos de anclaje. Se sabe de hace tiempo que la prote\u00edna tiene una regi\u00f3n peque\u00f1a, de s\u00f3lo 20 amino\u00e1cidos, que es clave para la supervivencia de las c\u00e9lulas tumorales.<\/p>\n<p>Ahora, el trabajo describe por primera vez que esta regi\u00f3n -habitualmente sin estructura y por tanto\u00a0a priori\u00a0descartada para enviar f\u00e1rmacos- toma una estructura en forma de h\u00e9lice. Al ganar esta h\u00e9lice -que no se entiende a\u00fan c\u00f3mo se produce-, otra prote\u00edna, llamada TFIIF, se engancha.\u00a0El estudio \u00a0evidencia que dicha interacci\u00f3n promueve la actividad del receptor de andr\u00f3genos y, consiguientemente, asegurar\u00eda la supervivencia y multiplicaci\u00f3n de las c\u00e9lulas tumorales.<br \/>\n\u00a0<\/p>\n<p><strong>\u25ba M\u00e1s informaci\u00f3n en la web del\u00a0<a href=\"https:\/\/www.irbbarcelona.org\/es\/news\/cerco-al-cancer-de-prostata-avanzado\" target=\"_blank\" rel=\"noopener noreferrer\">IRB Barcelona [+]<\/a><\/strong><\/p>\n<p><strong>\u25ba Art\u00edculo\u00a0de referencia:<\/strong><\/p>\n<p>Eva De Mol, Elzbieta Szulc, Claudio Di Sanza, Paula Mart\u00ednez-Crist\u00f3bal, Carlos W. Bertoncini, R. Bryn Fenwick, Marta Frigol\u00e9-Vivas, Marianela Mas\u00edn, Irene Hunter, V\u00edctor Buz\u00f3n, Isabelle Brun-Heath, Jes\u00fas Garc\u00eda, Gianni De Fabritiis, Eva Est\u00e9banez-Perpi\u00f1\u00e1, Iain J. McEwan, \u00c1ngel R. Nebreda, and Xavier Salvatella.<a href=\"http:\/\/linkinghub.elsevier.com\/retrieve\/pii\/S096921261730360X\" target=\"_blank\" rel=\"noopener noreferrer\"> <em>\u00abRegulation of androgen receptor activity by transient interactions of its transactivation domain with general transcription regulators\u00bb<\/em><\/a>. Structure\u00a0(2017).\u00a0DOI:\u00a0http:\/\/dx.doi.org\/10.1016\/j.str.2017.11.007<\/p>\n","protected":false},"excerpt":{"rendered":"<p>Un equipo liderado por el investigador ICREA en el <a href=\"http:\/\/www.pcb.ub.edu\/portal\/es\/cerca?p_p_id=cercador_WAR_empleatsempresesportlet&amp;p_p_lifecycle=0&amp;p_p_state=maximized&amp;p_p_mode=view&amp;p_p_col_id=column-1&amp;p_p_col_count=1&amp;_cercador_WAR_empleatsempresesportlet_jspPage=%2Fhtml%2Fcommon%2Fdetall-empresa.jsp&amp;_cercador_WAR_empleatsempresesportlet_empresaId=ENT_000001&amp;_cercador_WAR_empleatsempresesportlet_redirect=%2Fportal%2Fca%2Fcerca%3Fp_p_id%3Dcercador_WAR_empleatsempresesportlet%26p_p_lifecycle%3D0%26p_p_mode%3Dview%26_cercador_WAR_empleatsempresesportlet_keywords%3Dirb%26_cercador_WAR_empleatsempresesportlet_tab%3D1\" target=\"_blank\" rel=\"noopener noreferrer\">Instituto de Investigaci\u00f3n Biom\u00e9dica (IRB Barcelona<\/a>) en el Parc Cient\u00edfic de Barcelona,\u00a0Xavier Salvatella, ha descubierto un nuevo frente por donde atacar las c\u00e9lulas tumorales de pr\u00f3stata que han desarrollado resistencia al medicamento. El trabajo \u2013 publicado en la revista\u00a0Structure, del grupo\u00a0Cell\u2013\u00a0ha contado\u00a0con la colaboraci\u00f3n del laboratorio de Angel R. Nebreda\u00a0y del Laboratorio de Bioinform\u00e1tica Experimental, ambos\u00a0del IRB Barcelona, y de la Universidad de Barcelona.<\/p>\n<p>\u00a0<\/p>\n","protected":false},"author":1,"featured_media":27159,"comment_status":"closed","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"_acf_changed":false,"inline_featured_image":false,"footnotes":""},"categories":[9],"tags":[],"class_list":["post-39176","post","type-post","status-publish","format-standard","has-post-thumbnail","category-sin-categorizar"],"acf":[],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v28.0 - https:\/\/yoast.com\/product\/yoast-seo-wordpress\/ -->\n<title>Cerco al c\u00e1ncer de pr\u00f3stata avanzado - Parc Cient\u00edfic de Barcelona<\/title>\n<meta name=\"robots\" content=\"index, follow, max-snippet:-1, max-image-preview:large, max-video-preview:-1\" \/>\n<link rel=\"canonical\" href=\"https:\/\/www.pcb.ub.edu\/es\/cerco-al-cancer-de-prostata-avanzado\/\" \/>\n<meta property=\"og:locale\" content=\"es_ES\" \/>\n<meta property=\"og:type\" content=\"article\" \/>\n<meta property=\"og:title\" content=\"Cerco al c\u00e1ncer de pr\u00f3stata avanzado - Parc Cient\u00edfic de Barcelona\" \/>\n<meta property=\"og:description\" content=\"Un equipo liderado por el investigador ICREA en el Instituto de Investigaci\u00f3n Biom\u00e9dica (IRB Barcelona) en el Parc Cient\u00edfic de Barcelona,\u00a0Xavier Salvatella, ha descubierto un nuevo frente por donde atacar las c\u00e9lulas tumorales de pr\u00f3stata que han desarrollado resistencia al medicamento. El trabajo \u2013 publicado en la revista\u00a0Structure, del grupo\u00a0Cell\u2013\u00a0ha contado\u00a0con la colaboraci\u00f3n del laboratorio de Angel R. 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