Publications

"Synthesis of a Targeted Library of Potential Tryptase Inhibitors" M. García, X. del Rio, S. Silvestre, M. Rubiralta, V. Segarra, E. Loyoza, A. Diez. Org. & Biol. Chem., 2004, 2, 1633-1642.

"Constrained derivatives of stylostatin 1. Part 1. Synthesis and biological evaluation as potential anticancer agents" P. Forns, J. Piró, C. Cuevas, M. García, M. Rubiralta, E. Giralt, A. Diez. J. Med. Chem., 2003, 46, 5825-5833.

"Synthesis of 3-aminolactams as X-Gly constrained pseudodipeptides and conformational study of the Trp-Gly surrogate" M. Ecija, M.J. Kogan, M. Rubiralta, E. Giralt, A. Diez, N. Casamitjana. J. Org. Chem, 2003, 68, 9541-9553.

"Complete 1H and 13C NMR chemical shift assignment of N1- and N3-alkyl nitrohistidines and of 1,4,6,7-tetrahydroimidazo[4,5-b]pyridines" C. Escolano, M. J. Kogan, M. Rubiralta, E. Giralt, A. Diez. Magnetic Resonance in Chemistry, 2003, 41, 219-222.

"Spirolactams as Conformationally Restricted Pseudopeptides: Synthesis and Conformational Analysis" M.M. Fernández, A. Diez, M. Rubiralta, E. Montenegro, N. Casamitjana, M. J. Kogan, E. Giralt. J. Org. Chem., 2002, 67, 7587-7599.

"Spirolactams as Conformationally Restricted Pseudopeptides: Synthesis and Conformational Analysis" M.M. Fernández, A. Diez, M. Rubiralta, E. Montenegro, N. Casamitjana, M. J. Kogan, E. Giralt. J. Org. Chem., 2002, 67, 7587-7599.

"Synthesis of Constrained Pseudopeptides by Regioselective Ring Opening of 3,4-Aziridinopiperidin-2-ones" J. Piró, P. Forns, J. Blanchet, M. Bonin, L. Micouin, A. Diez. Tetrahedron: Asymm., 2002, 13, 995-1004.

"Synthesis and Structural Study of 6-Amino-1,4,6,7-tetrahydroimidazo[4,5-b]pyridin-5-ones" C. Escolano, M. Rubiralta, A. Diez. Tetrahedron Letters, 2002, 43, 4343-4346.

"Aminoimidazo[1,2-a]pyridines: regioselective synthesis of substituted imidazonaphthyridines, azacarbolines and cyclazines" Chezal, Jean M.; Moreau, Emmanuel; Chavignon, Olivier; Gaumet, Vincent; Metin, Jacques; Blache, Yves; Diez, Anna; Fradera, Xavier; Luque, Javier; Teulade, Jean C. Tetrahedron, 2002, 58, 295-307.

"Piperidones: from Alkaloids to Pseudopeptides" P. Forns, M. Rubiralta, A. Diez. Contibutions to Science, 2001, 2, 63-86.

"Solid Phase Synthesis of Polyhydroxylactams" J. Piró, M. Rubiralta, E. Giralt, A. Diez. Tetrahedron Lett., 2001, 42, 871-873.

"Synthesis of a 3-Aminopiperidin-2,5-dione as a Conformationally Constrained Surrogate of the Ala-Gly Dipeptide" M. A. Estiarte, A. Diez, M. Rubiralta, R.F.W. Jackson. Tetrahedron, 2001, 57, 157-161.

"Absolute Configuration of a C2 Symmetric bis-Thiophenol" R.B. Bates, M. D. Carducci, A. Diez, P. Forns, V.V. Kane, M. Rubiralta. Acta Cryst., 2000, C56, e484.

"Oxazolopiperidin-2-ones as Type II' beta-Turn Mimetics: Synthesis and Conformational Analysis" M.A. Estiarte, M. Rubiralta, A. Diez, M. Thormann, E. Giralt. J. Org. Chem., 2000, 65, 6992-6999.

"New Efficient Method for the Synthesis of 4-Hydroxynorvaline" M. García, A. Serra, M. Rubiralta, A. Diez, V. Segarra, H. Ryder, E. Lozoya, J.M. Palacios. Tetrahedron: Asymmetry, 2000, 11, 991-994.

"3-Amino-2-piperidones as Constrained Pseudopeptides: Preparation of a New Ser-Leu Surrogate" J. Piró, M. Rubiralta, E. Giralt, A. Diez. Tetrahedron Letters, 1999, 40, 4865-4868.

"Synthesis and Synthetic Applications of 3-Amino-D5-piperidein-2-ones: Synthesis of Methionine-derived Pseudopeptides" M.A. Estiarte, M. de Souza, X. del Río, R. H. Dodd, M. Rubiralta, A. Diez Tetrahedron, 1999, 55, 10173-10186.

"Methylenation and Oxidation of Chiral Non-Racemic 2-Piperidones. Reactivity of a New 3-Oxolactam" P. Forns, M. Fernández, A. Diez, M. Rubiralta, M.-P. Cherrier, M. Bonin, J.-C. Quirion. Synthesis, 1999, 258-263.